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{{Adrenergic receptor modulators}} {{Dopamine receptor modulators}} ...

...k IN | title = The anorectic effect of SK&F 38393, a selective dopamine D1 receptor agonist: a microstructural analysis of feeding and related behaviour | jour {{Dopamine receptor modulators}} ...

...th either minimal or negligible effects on the [[D2 receptor|D₂ receptor]]. ...CNS Drug Reviews | title=SCH 23390: The First Selective Dopamine D 1 ‐Like Receptor Antagonist | volume=7 | issue=4 | pages=399–414 | date= December 2001 | doi ...

{{Adrenergic receptor modulators}} {{Dopamine receptor modulators}} ...

! Receptor !! K_i (nM) !! Notes | [[5-HT1A receptor|5-HT_1A]] || 17.3 || ...

...not used therapeutically as a [[neuroleptic]] because it does not block [[dopamine receptors]] well.{{Citation needed|date=July 2022}} .../sub>-adrenergic receptor]], and [[histamine]] [[H1 receptor|H₁ receptor]].{{Citation needed|date=July 2022}} ...

..., Dutertre M, Smith CL | title = SKF-82958 is a subtype-selective estrogen receptor-alpha (ERalpha ) agonist that induces functional interactions between ERalp {{Dopamine receptor modulators}} ...

...cts in the rat of dihydrexidine, a high-potency, full-efficacy D1 dopamine receptor agonist. | journal = Neuropsychopharmacology | volume = 5 | issue = 3 | pag ...ols DE, Mailman RB, George MS | title = A single 20 mg dose of the full D1 dopamine agonist dihydrexidine (DAR-0100) increases prefrontal perfusion in schizoph ...

...all TCAs, TeCAs have only low affinity for the [[muscarinic acetylcholine receptor]]s, and for this reason, are associated with few or no [[anticholinergic]] ...y constant}}, {{abbr|nM|nanomolar}}) for various [[receptor (biochemistry)|receptor]]s and [[membrane transport protein|transporter]]s are as follows:<ref name ...

...display-authors = 6 | title = Muscarinic receptor agonists, like dopamine receptor antagonist antipsychotics, inhibit conditioned avoidance response in rats | {{Muscarinic acetylcholine receptor modulators}} ...

...(psychology)|mood]] regulation,<ref name="Julien2004" /> notably [[5-HT1A receptor|5-HT_1A]]-mediated transmission.<ref name="HalesShahrokh2009">{{c ...e A, Brocco M, Loiseau F, etal | title = S32212, a novel serotonin type 2C receptor inverse agonist/α2-adrenoceptor antagonist and potential antidepressant: II ...

{{Short description|Dopamine agonist medication}} ...yons KE | title = Transdermal rotigotine: a clinically innovative dopamine-receptor agonist for the management of Parkinson's disease | journal = Pharmacothera ...

...s T, Harp J, Budygin E, Jones S | title = Diphenylpyraline, a histamine H1 receptor antagonist, has psychostimulant properties | journal = Eur J Pharmacol | vo {{Acetylcholine receptor modulators}} ...

{{Adrenergic receptor modulators}} {{Dopamine receptor modulators}} ...

{{Adrenergic receptor modulators}} {{Dopamine receptor modulators}} ...

...t]] and also has high [[affinity (pharmacology)|affinity]] for the [[sigma receptor]], possibly playing a role in its atypical neuroleptic action.<ref name="pm {{Dopamine receptor modulators}} ...

..., Yuan H, Myers SJ, Dingledine R | display-authors = 6 | title = Glutamate receptor ion channels: structure, regulation, and function | journal = Pharmacologic ...NQX-induced toxicity in cultured rat hippocampal neurons: an apparent AMPA receptor-independent effect? | journal = Neurochemistry International | volume = 42 ...

...of beta-carbolines and related agents at serotonin (5-HT(2) and 5-HT(1A)), dopamine (D(2)) and benzodiazepine receptors | journal = Drug Alcohol Depend | volum {{Monoamine metabolism modulators}} ...

...pmid12808385">{{cite journal | vauthors = Bankowski BJ, Zacur HA | title = Dopamine agonist therapy for hyperprolactinemia | journal = Clinical Obstetrics and ...itle = Ergocryptine and other ergot alkaloids stimulate the release of [3H]dopamine from rat striatal synaptosomes | journal = Journal of Animal Science | volu ...

...[[5-HT6 receptor|5-HT₆]], and [[5-HT7 receptor|5-HT₇ receptor]]s.<ref name=PDSP>{{cite web|title=PDSD Ki Database |date=12 January 2011 | ! Macromolecule (Receptor or transporter protein) !! K_i [nM]<ref name = PDSP/> ...