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- ...] and [[TAAR5]] with similar [[potency (pharmacology)|potency]] as for the TAAR1 (all in the case of the human proteins).<ref name="KhanNawaz2016" /><ref na ...s relationship is not typical of the [[endocrine system]], indicating that TAAR1 activity may not be coupled to [[G protein]]s in some [[tissue (biology)|ti ...12 KB (1,643 words) - 12:47, 13 April 2025
- ...inity (K<sub>i</sub>) of 3,100{{nbsp}}nM and was not assessed at the human TAAR1.<ref name="KolaczynskaLuethiTrachsel2019" /> {{Serotonin receptor modulators}} ...20 KB (2,383 words) - 23:08, 17 June 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || 4,100 (K<sub>i</sub>) (mouse)<br />1 ...mine-associated receptor 1]] (TAAR1), but only weak affinity for the mouse TAAR1.<ref name="Gil-MartinsBarbosaBorges2025" /><ref name="RickliLuethiReinisch2 ...21 KB (2,745 words) - 19:49, 29 May 2025
- ...M and 3,200{{nbsp}}nM, respectively), whereas it was inactive at the human TAAR1 ({{Abbr|EC<sub>50</sub>|half-maximal effective concentration}} > 10,000{{nb {{Serotonin receptor modulators}} ...21 KB (2,522 words) - 03:16, 8 June 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || 3,500 (K<sub>i</sub>) (mouse)<br />1 {{Serotonin receptor modulators}} ...20 KB (2,582 words) - 19:49, 29 May 2025
- ...analog|analogue]]s might enhance their effects relative to MRAs possessing TAAR1 agonism.<ref name="MaierMayerBrandt2018" /><ref name="MaierMayerLuethi2018" {{Serotonin receptor modulators}} ...28 KB (3,491 words) - 19:00, 23 May 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || 280 (K<sub>i</sub>) (mouse)<br />20 ...iated receptor 1]] (TAAR1) and lower but still high affinity for the mouse TAAR1.<ref name="RickliLuethiReinisch2015" /> ...26 KB (3,493 words) - 22:27, 20 June 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || 2,337–4,500 (K<sub>i</sub>) (mouse)< {{Serotonin receptor modulators}} ...18 KB (2,382 words) - 19:49, 29 May 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || >20,000 (K<sub>i</sub>) (mouse)<br / {{Serotonin receptor modulators}} ...17 KB (2,208 words) - 00:39, 21 June 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || >15,000 (K<sub>i</sub>) (mouse)<br / ...t interact with the rodent or human [[trace amine-associated receptor 1]] (TAAR1).<ref name="SimmlerBuchyChaboz2016" /> ...19 KB (2,415 words) - 23:57, 9 May 2025
- ...uropharm.2013.11.008 | url = }}</ref> However, it is inactive at the human TAAR1 ({{Abbrlink|EC<sub>50</sub>|half-maximal effective concentration}} > 10,000 {{Serotonin receptor modulators}} ...24 KB (3,174 words) - 00:01, 10 May 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || 2,200 (K<sub>i</sub>) (mouse)<br />4 {{Serotonin receptor modulators}} ...24 KB (3,055 words) - 16:28, 16 June 2025
- ====Dopamine receptor positive allosteric modulators==== ====Dopamine receptor negative allosteric modulators==== ...28 KB (3,342 words) - 13:26, 17 June 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || 3,300 (K<sub>i</sub>) (mouse)<br />1 {{Serotonin receptor modulators}} ...23 KB (2,974 words) - 03:13, 10 June 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || {{Abbr|ND|No data}} {{Serotonin receptor modulators}} ...20 KB (2,622 words) - 19:52, 23 June 2025
- ...iagram">{{cite book | vauthors = Beardsley PM, Hauser KF | chapter = Glial Modulators as Potential Treatments of Psychostimulant Abuse | title = Emerging Targets ...amate clearance abilities. Furthermore, molecular alterations in astrocyte TAAR1 levels correspond to changes in astrocyte EAAT-2 levels and function. | pmc ...24 KB (3,219 words) - 15:14, 24 September 2023
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || >15,000 (K<sub>i</sub>) (mouse)<br / ...iochemistry)|ligand]] of the rodent [[trace amine-associated receptor 1]] (TAAR1).<ref name="RickliMoningHoener2016" /><ref name="SimmlerBuchyChaboz2016" /> ...19 KB (2,482 words) - 00:30, 15 May 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || 710 (K<sub>i</sub>) (mouse)<br />30 {{Serotonin receptor modulators}} ...25 KB (3,258 words) - 01:38, 1 June 2025
- ...ssociated receptor 1]] (TAAR1) and a weak agonist of the [[rhesus monkey]] TAAR1.<ref name="LewinMillerGilmour2011">{{cite journal | vauthors = Lewin AH, Mi {{Serotonin receptor modulators}} ...28 KB (3,407 words) - 12:33, 25 May 2025
- | {{Abbrlink|TAAR1|Trace amine-associated receptor 1}} || 1,200 (K<sub>i</sub>) (mouse)<br />6 {{Serotonin receptor modulators}} ...26 KB (3,357 words) - 19:49, 29 May 2025