Neuropeptide Y receptor Y1
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Template:Short description Template:Infobox gene Neuropeptide Y receptor type 1 is a protein that in humans is encoded by the NPY1R gene.[1][2]
Selective ligands
Agonists
- Neuropeptide Y (endogenous agonist, non subtype selective)
- Peptide YY
Antagonists
- Peptide
- BVD-10 (selective NPY1 antagonist, CAS# 262418-00-8)
- GR-231,118 (mixed NPY1 antagonist / NPY4 agonist, CAS# 158859-98-4)
- Non-peptide
- BIBO-3304 (CAS# 191868-14-1)
- BIBP-3226 (CAS# 159013-54-4)
- PD-160,170 (CAS# 181468-88-2)
Available Structures
- 5ZBH (Neuropeptide Y1 bound to antagonist BMS-193835)[3]
- 5ZBQ (Neuropeptide Y1 bound to antagonist UR-MK299)[3]
See also
References
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Further reading
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External links
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- Template:PDBe-KB2
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