Glibornuride

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Glibornuride
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MeSH C073323
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Molar mass 366.48 g/mol
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Glibornuride (INN) is an anti-diabetic drug from the group of sulfonylureas.[1] It is manufactured by MEDA Pharma and sold in Switzerland under the brand name Glutril.[2]

Synthesis

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Glibornuride synthesis:[3] See also: U.S. patent 3770761; eidem, U.S. patent 3654357 (to Hoffmann-La Roche).

Gliburnide is an endo-endo derivative made from camphor-3-carboxamide by borohydride reduction (exo approach), followed by Hofmann rearrangement to carbamate, followed by displacement with sodium tosylamide.

References

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