Exatecan

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Exatecan is a drug which is a structural analog of camptothecin with antineoplastic activity.[1]

A derivative is used in Trastuzumab deruxtecan.

Synthesis

File:Exatecan scheme.png
Exatecan synthesis[2]

References

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  2. H. Terasawa, A. Ejima, S. Ohsuki, K. Uoto, U.S. Patent 5,834,476 (1998).

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