Bisulepin
Jump to navigation
Jump to search
Template:Short description Template:Drugbox
Bisulepin is strong and relatively selective antihistamine (H1 antagonist) with hypnotic, antiadrenergic and very weak anticholinergic and antiserotonergic effects. Bisulepin is marketed in the Czech Republic and Slovakia under the trademark Dithiaden as tablets and injections.
The registered active form is the trans- (i.e. E-) isomer.[1][2]
See also
References
- ↑ Script error: No such module "Citation/CS1".
- ↑ Pharmacopoea Bohemoslovenica 4 (1987), vol. 2, p. 132 states that Bisulepinium chloratum (bisulepinium chloride) is trans-[3-(4,9-dihydro-thieno[2,3-c][2]benzithiepin-4-yliden)propyl]dimethylamoniumchlorid (Czech). The cis- isomer is considered as an impurity, max. amount 2.0 %.
External links
Script error: No such module "Navbox".