Ajmalan

From Wikipedia, the free encyclopedia
Jump to navigation Jump to search

<templatestyles src="Chembox/styles.css"/>

Template:Chembox image cellTemplate:Chembox AllOtherNamesTemplate:Chembox headerbarTemplate:Chembox IndexlistTemplate:Chembox JmolTemplate:Chembox ChEMBLTemplate:Chembox ECHATemplate:Chembox E numberTemplate:Chembox IUPHAR ligandTemplate:Chembox UNIITemplate:Chembox CompToxTemplate:Chembox Datapage checkTemplate:Yesno
Ajmalan
Template:Longitem Template:Unbulleted list
ChEBI Template:Unbulleted list
ChemSpider Template:Unbulleted list
DrugBank Template:Unbulleted list
EC Number Template:Unbulleted list
KEGG Template:Unbulleted list
Template:Longitem Template:Unbulleted list
RTECS number Template:Unbulleted list
Script error: No such module "collapsible list".
Script error: No such module "collapsible list".

Template:Chembox Footer/tracking container onlyScript error: No such module "TemplatePar".Template:Short description

Ajmalan is a parent hydride used in the IUPAC nomenclature of natural products and also in CAS nomenclature.[1] It is a 20-carbon alkaloid with six rings and seven chiral centres.

The name is derived from ajmaline, an antiarrhythmic alkaloid isolated from the roots of Rauvolfia serpentina[2] which is formally a dihydroxy-derivative of ajmalan. The –an ending indicates that ajmalan is partially saturated. Ajmaline itself is named after Hakim Ajmal Khan, a distinguished practitioner of the Unani school of traditional medicine in South Asia.[3]

The absolute configuration of the seven chiral carbon atoms in ajmalan is defined by convention, as is the numbering system.[1] The stereochemistry is the same as that in naturally occurring ajmaline, and corresponds to (2R,3S,5S,7S,15S,16R,20S) using conventional numbering.

Ajmalan can be systematically named as

Template:Chem name

or as

Template:Chem name.

Note that the numbering of the atoms in the systematic names is different from the conventional numbering of ajmalan.[4]

The ajmalan skeleton is similar to those of certain other alkaloids, and ajmalan could also be given the following semisystematic names:

Template:Chem name
(2β,5β,7β,16R,20β)-1-methyl-2,7-dihydro-5,16:7,17-dicyclocorynan;
(2β,7β,16R,20β)-1-methyl-2,7,19,20-tetrahydro-7,17-cyclosarpagan;
(2β,3α,7β,20β)-1-methyl-2,7,19,20-tetrahydro-3,4:7,17-dicyclo-22-norvobasan;
(2β,5β,7β,16R,20β)-1-methyl-2,7-dihydro-5,16:7,17-dicyclo-17-secoyohimban.

However, the relative complexity even of these names justifies the use of ajmalan as a defined parent hydride in alkaloid nomenclature.

References

<templatestyles src="Reflist/styles.css" />

  1. a b Template:IUPAC natural products 1999.
  2. Siddiqui, S.; Siddiqui, R. H. (1931). J. Indian Chem. Soc. 8: 667–80.
  3. Ahmed Nasim Sandilvi (2003). "Salimuzzaman Siddiqui: pioneer of scientific research in Pakistan. Template:Webarchive" Daily Dawn, 2003-04-12. Retrieved on 2007-07-19.
  4. The numbering is also different between the von Baeyer name and the fusion name, given the different conventions which apply to the two methods of nomenclature.

Script error: No such module "Check for unknown parameters".