ABCC4
Template:Short description Template:Infobox gene ATP-binding cassette sub-family C member 4 (ABCC4), also known as the multidrug resistance-associated protein 4 (MRP4) or multi-specific organic anion transporter B (MOAT-B), is a protein that in humans is encoded by the ABCC4 gene.[1][2]
ABCC4 acts as a regulator of intracellular cyclic nucleotide levels and as a mediator of cAMP-dependent signal transduction to the nucleus.[3] MRP4/ABCC4 also transports prostaglandins, for example PGE2, out of the cell where they can bind receptors.[4]
MRP4/ABCC4 expression is dysregulated in several cancers [5][6][7] and is also upregulated in peritoneal endometriosis.[8]
Interactive pathway map
Template:FluoropyrimidineActivity WP1601
See also
References
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- ↑ Holla VR, Backlund MG, Yang P, Newman RA, DuBois RN. Regulation of prostaglandin transporters in colorectalneoplasia. Cancer Prev Res (Phila). 2008;1(2) 93-9.
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Further reading
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