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==List of nonsteroidal steroid receptor modulators== * {{abbrlink|SERMs|Selective estrogen receptor modulators}}: [[acolbifene]], [[afimoxifene]], [[arzoxifene]], [[bazedoxifene]], [[bro ...

{{ATC codes lead|G|03|Sex hormones and modulators of the genital system|vet=add}} :G03DA04 [[Progesterone (medication)|Progesterone]] ...

...mmended to induce bleeding on a regular schedule. [[Selective progesterone receptor modulator]]s (SPRMs) are sometimes used to stop uterine bleeding.<ref name= ...

...SH number|D06.347.360|Estrogen+Receptor+Modulators}} – [[estrogen receptor modulators]]==== ...7|Selective+Estrogen+Receptor+Modulators}} – [[selective estrogen receptor modulators]] ...

{{Short description|Cytoplasmic receptor protein found inside cells}} ...is a protein found inside cells. It is activated by the steroid hormone [[progesterone]]. ...

| Name = ERG2/Sigma-1 receptor |Name=Sigma intracellular receptor 2 ...

{{Short description|Nuclear receptor that mediates the effects of the mineralocorticoid hormone Aldosterone}} ...ley LL, Henry WM, Nowak NJ, Shows TB | title = The human mineralocorticoid receptor gene (MLR) is located on chromosome 4 at q31.2 | journal = Cytogenetics and ...

| Caption = [[Ulipristal acetate]], an {{abbr|SPRM|selective progesterone receptor modulator}} that is used as an [[emergency contraceptive]] and in the treat | Biological_target = [[Progesterone receptor]] ...

...tion to the PR and AR, gestrinone has been found to bind to the [[estrogen receptor]] (ER) with relatively "avid" affinity.<ref name="pmid3490730">{{cite journ ...{{abbrlink|GR|Glucocorticoid receptor}} || {{abbrlink|MR|Mineralocorticoid receptor}} || {{abbrlink|SHBG|Sex hormone-binding globulin}} || {{abbrlink|CBG|Corti ...

...d H, Blomquist P, Berkenstam A | title = Identification of a human nuclear receptor defines a new signaling pathway for CYP3A induction | journal = Proceedings ...70465"/><ref name="entrez">{{cite web | title = Entrez Gene: NR1I2 nuclear receptor subfamily 1, group I, member 2| url = https://www.ncbi.nlm.nih.gov/sites/en ...

..., Bittman R, Hurley S, Kleiman J, Gatlin M, Pitt B | title = Eplerenone, a Selective Aldosterone Blocker, in Patients with Left Ventricular Dysfunction after My ...kman DL, Sing YL, Whelihan B | title = Eplerenone: a selective aldosterone receptor antagonist (SARA) | journal = Cardiovascular Drug Reviews | volume = 19 | i ...

...ay also exert effects on [[gene expression]] via nuclear [[steroid hormone receptor]]s. Neurosteroids have a wide range of potential clinical applications from ...[positive allosteric modulator]]s of the [[GABAA receptor|GABA_A receptor]] (especially [[GABRD|δ subunit]]-containing [[isoform]]s), and possess, in ...

| Name = [[estrogen receptor alpha|estrogen receptor 1]] (ER-alpha) | Symbol = [[estrogen receptor alpha|ESR1]] ...

{{Short description|Drugs acting on the estrogen receptor}} | Synonyms = SERM; Estrogen receptor agonist/antagonist; ERAA ...

....<ref>{{cite journal | vauthors = Serock MR, Wells AK, Khalil RA | title = Modulators of vascular sex hormone receptors and their effects in estrogen-deficiency ...(''Dioscorea villosa'') extract creams are not effective since the natural progesterone present in the extract is not bioavailable.<ref>{{cite web | author = Harva ...

...eceptor|estrogen]], [[progesterone receptor|progesterone]], and [[androgen receptor]]s.<ref name="Cano2017">{{cite book | vauthors = Cano A | title = Menopause ...bserved with most of the [[aromatase inhibitor]]s and [[selective estrogen receptor modulator]]s that were included in the analysis.<ref name="pmid26582062" /> ...

...3–}}</ref> These include direct binding to and activation of [[sex hormone receptor]]s, direct [[enzyme inhibitor|inhibition]] of [[enzyme]]s involved in [[ste ...oassay, indicating that it could be regarded as a [[selective progesterone receptor modulator]] (SPRM).<ref name="ThomasRock2012" /> Although the [[affinity (p ...

...nd to double stranded [[DNA]] (magenta) and two molecules of the [[Nuclear receptor coactivator 2|NCOA2]] coactivator (red). The PPAR-γ antagonist GW9662 and R ...rmone]]s, [[vitamins]], and certain other molecules. These intracellular [[receptor (biochemistry)|receptors]] work with other proteins to regulate the [[gene ...

| class = [[Selective estrogen receptor modulator]]; [[Progonadotropin]] ...–386 }}</ref><ref name=FDAlabel/> Clomifene is in the [[selective estrogen receptor modulator]] (SERM) family of medication and is a nonsteroidal medication.<r ...

...[progesterone receptor]], the [[biological target]] of progestogens like [[progesterone]].<ref name="pmid8616978" /><ref name="pmid8808163" /> It has very weak [[a Desogestrel is a hormone blocker, [[progesterone]] receptors [[agonist]], and [[antiandrogen]]. It is used in conjunction wi ...