5-HT1F receptor
(Redirected from 5-HT1F)
Template:Infobox gene 5-hydroxytryptamine (serotonin) receptor 1F, also known as HTR1F is a 5-HT1 receptor protein and also denotes the human gene encoding it.[1][2][3][4][5]
Agonists
- 5-n-Butyryloxy-DMT:[6] >60-fold selectivity versus 5-HT1E receptor
- BRL-54443 - mixed 5-HT1E/1F agonist
- Eletriptan - mixed 5-HT1B/1D/1E/1F/2B/7 agonist
- LY-334,370[7] - as well as related benzamides[8]
- LY-344,864 (N-[(3R)-3-(Dimethylamino)-2,3,4,9-tetrahydro-1H-carbazol-6-yl]-4-fluorobenzamide)
- Naratriptan - mixed 5-HT1B/1D/1F agonist
- Lasmiditan - selective 5-HT1F agonist, a first-in-class ditan molecule
Antagonists
MLS000756415[9]
See also
References
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- ↑ PubChem: MLS000756415
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Further reading
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External links
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- Template:UCSC gene info
This article incorporates text from the United States National Library of Medicine, which is in the public domain.
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Template:Serotonergics