Fludiazepam
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Fludiazepam,[1] marketed under the brand name Erispan (エリスパン)[2][3] is a potent benzodiazepine and 2ʹ-fluoro derivative of diazepam,[4] originally developed by Hoffmann-La Roche in the 1960s.[5] It is marketed in Japan and Taiwan. Script error: No such module "Unsubst". It exerts its pharmacological properties via enhancement of GABAergic inhibition.[6] Fludiazepam has 4 times more binding affinity for benzodiazepine receptors than diazepam.[7] It possesses anxiolytic,[8][9][10] anticonvulsant, sedative, hypnotic and skeletal muscle relaxant properties.[11] Fludiazepam has been used recreationally.[12]
See also
- Diazepam
- Diclazepam (the 2ʹ-chloro analog)
- Difludiazepam (the 2',6'-difluoro derivative)
- Flunitrazepam (the 7-nitro analog)
- Flualprazolam (the triazolo derivative)
- Ro20-8552
References
External links
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- Template:In lang Official Dainippon Sumitomo Pharma Website Template:Webarchive
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- ↑ US Patent 3371085 5-aryl-3h-1,4-benzodiazepin-2(1h)-ones
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- ↑ US Patent 3299053 -ARYL-JH-L,X-BENZODIAZEPIN-Z(LH)-ONES
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